Thierry BESSON

Professeur Chimie Thérapeutique / Professor (Full) in Medicinal Chemistry

University of Rouen

France

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Thierry BESSON is a Full Professor in Medicinal Chemistry at Université de Rouen Normandie UFR Santé, France. His research focuses on medicinal chemistry, with recent articles exploring the synthesis and biological evaluation of novel compounds, including DYRK1A inhibitors for Down syndrome acute lymphoblastic leukemia, and multitarget ligands for Alzheimer's disease. His work also includes advancements in the synthesis of various thiazole-fused compounds and the development of dual inhibitors for kinase targets.

Thierry BESSON

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Articles (15)

Efficacy of DYRK1A inhibitors in novel models of Down syndrome acute lymphoblastic leukemia

Synthesis of Thiazole-fused Tricyclic Quinazolinone Alkaloids and Their Derivatives

Contribution of Professor Charles W. Rees to the development of the chemistry of disulfur dichloride

Design, synthesis and preliminary biological evaluation of rivastigmine-INDY hybrids as multitarget ligands against Alzheimer's disease by targeting butyrylcholinesterase and DYRK1A/CLK1 kinases

Novel Thiazole-Fused [4,5-g] or [5,4-g]Quinazolin-8-ones and Their Quinazoline Analogues: Synthesis and Biological Evaluation

Synthesis of Trifunctional Thiazole-Fused Anthranilonitrile and Anthranilic Acid Derivatives

Photocatalyst-Free, Visible-Light-Mediated C–H Perfluoroalkylation of Quinazolin-4(3H)-ones with perfluoroalkyl Iodides

Straightforward Access to a New Class of Dual DYRK1A/CLK1 Inhibitors Possessing a Simple Dihydroquinoline Core

Synthesis of 2-Cyanobenzothiazoles via Pd-Catalyzed/Cu-Assisted C-H Functionalization/Intramolecular C-S Bond Formation from N-Arylcyanothioformamides

Monitoring of Catalyst-Free Microwave-Assisted MCR-Type Synthesis of 2-Amino-3-cyano-4H-chromene Derivatives Using Raman Spectrometry

Relieving DYRK1A repression of MKL1 confers an adult-like phenotype to human infantile megakaryocytes

Review on the Synthesis and Therapeutic Potential of Pyrido[2,3-d], [3,2-d], [3,4-d] and [4,3-d]pyrimidine Derivatives

A skills framework integrating professionally relevant medicinal chemistry proficiencies to strengthen the contemporary practice of pharmacy

Recent Advances in Transition-Metal-Free Late-Stage C-H and N-H Arylation of Heteroarenes Using Diaryliodonium Salts

Microwave-Assisted Sequential One-Pot Synthesis of 8-Substituted Pyrazolo[1,5-a][1,3,5]triazines

Collaborators (6)

Jana Sopkova-de Oliveira Santos

Marc Pudlo

Camelia Iancu-Rubin

Laurence C Cheung

Line Bourel

Sabine Berteina-Raboin

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