Steffen Pockes

University of Regensburg

Germany

This profile is automatically generated from trusted academic sources.

Google Scholar

ORCID

How do I reach out?

Meet Kite AI

Contact this professor

ORCID

Google Scholar

Research Interests

Pharmacology

100%

Biochemistry

50%

G Protein-coupled Receptor

70%

Receptor Biology

60%

Neuropharmacology

50%

Ligand Design

40%

Apoptosis

40%

Ask ApplyKite AI

Start chatting

How can you help me contact this professor?

What are this professor's research interests?

How should I write an email to this professor?

Articles20

Activation of Multiple G Protein Pathways to Characterize the Five Dopamine Receptor Subtypes Using Bioluminescence Technology

Article Link

Year:

2024

Dual Piperidine-Based Histamine H3 and Sigma-1 Receptor Ligands in the Treatment of Nociceptive and Neuropathic Pain.

Article Link

Year:

2023

Ergometrine stimulates histamine H2 receptors in the isolated human atrium

Article Link

Year:

2023

Development of Fluorescent AF64394 Analogues Enables Real-Time Binding Studies for the Orphan Class A GPCR GPR3

Article Link

Year:

2023

Discovery of a Tritiated Radioligand with High Affinity and Selectivity for the Histamine H3 Receptor

Article Link

Year:

2023

Fluorescent Tools for the Imaging of Dopamine D2‐Like Receptors

Article Link

Year:

2023

Shedding Light on the D1‐Like Receptors: A Fluorescence‐Based Toolbox for Visualization of the D1 and D5 Receptors

Article Link

Year:

2023

An electrophilic fragment screening for the development of small molecules targeting caspase-2

Article Link

Year:

2023

Clonidine stimulates force of contraction via histamine H2 receptors in the human atrium

Article Link

Year:

2023

Lysergic acid diethylamide stimulates cardiac human H2 histamine and cardiac human 5-HT4-serotonin receptors

Article Link

Year:

2023

Characterization of caspase-2 inhibitors based on specific sites of caspase-2-mediated proteolysis

Article Link

Year:

2022

Structure-Based Design and Biological Evaluation of Novel Caspase-2 Inhibitors Based on the Peptide AcVDVAD-CHO and the Caspase-2-Mediated Tau Cleavage Sequence YKPVD314

Article Link

Year:

2022

Targeting caspase-2 interactions with tau in Alzheimer's disease and related dementias

Article Link

Year:

2022

Investigating the ligand agonism and antagonism at the D2long receptor by dynamic mass redistribution

Article Link

Year:

2022

Caspase-2 Inhibitor Blocks Tau Truncation and Restores Excitatory Neurotransmission in Neurons Modeling FTDP-17 Tauopathy

Article Link

Year:

2022

Structural and Molecular Insight into Piperazine and Piperidine Derivatives as Histamine H3 and Sigma-1 Receptor Antagonists with Promising Antinociceptive Properties.

Article Link

Year:

2021

Cardiac effects of novel histamine H2 receptor agonists

Article Link

Year:

2021

A Versatile Sub-Nanomolar Fluorescent Ligand Enables NanoBRET Binding Studies and Single-Molecule Microscopy at the Histamine H3 Receptor

Article Link

Year:

2021

Abolishing Dopamine D2long/D3 Receptor Affinity of Subtype-Selective Carbamoylguanidine-Type Histamine H2 Receptor Agonists

Article Link

Year:

2021

Histamine H2 receptor radioligands: triumphs and challenges

Article Link

Year:

2021

Collaborators5

Katarzyna Szczepańska

Institute of Pharmacology

POLAND

David Reiner-Link

Københavns Universitet

DENMARK

Enrique José Cobos Del Moral

Universidad de Granada

SPAIN

Barry Finzel

University of Minnesota

UNITED STATES

Ulrich Gergs

Martin Luther University Halle-Wittenberg

GERMANY

How do I reach out?

Meet Kite AI

Steffen Pockes

How do I reach out?

Contact this professor

Research Interests

Ask ApplyKite AI

Articles20

Activation of Multiple G Protein Pathways to Characterize the Five Dopamine Receptor Subtypes Using Bioluminescence Technology

Dual Piperidine-Based Histamine H<sub>3</sub> and Sigma-1 Receptor Ligands in the Treatment of Nociceptive and Neuropathic Pain.

Ergometrine stimulates histamine H2 receptors in the isolated human atrium

Development of Fluorescent AF64394 Analogues Enables Real-Time Binding Studies for the Orphan Class A GPCR GPR3

Discovery of a Tritiated Radioligand with High Affinity and Selectivity for the Histamine H<sub>3</sub> Receptor

Fluorescent Tools for the Imaging of Dopamine D2‐Like Receptors

Shedding Light on the D1‐Like Receptors: A Fluorescence‐Based Toolbox for Visualization of the D1 and D5 Receptors

An electrophilic fragment screening for the development of small molecules targeting caspase-2

Clonidine stimulates force of contraction via histamine H2 receptors in the human atrium

Lysergic acid diethylamide stimulates cardiac human H2 histamine and cardiac human 5-HT4-serotonin receptors

Characterization of caspase-2 inhibitors based on specific sites of caspase-2-mediated proteolysis

Structure-Based Design and Biological Evaluation of Novel Caspase-2 Inhibitors Based on the Peptide AcVDVAD-CHO and the Caspase-2-Mediated Tau Cleavage Sequence YKPVD314

Targeting caspase-2 interactions with tau in Alzheimer's disease and related dementias

Investigating the ligand agonism and antagonism at the D2long receptor by dynamic mass redistribution

Caspase-2 Inhibitor Blocks Tau Truncation and Restores Excitatory Neurotransmission in Neurons Modeling FTDP-17 Tauopathy

Structural and Molecular Insight into Piperazine and Piperidine Derivatives as Histamine H<sub>3</sub> and Sigma-1 Receptor Antagonists with Promising Antinociceptive Properties.

Cardiac effects of novel histamine H2 receptor agonists

A Versatile Sub-Nanomolar Fluorescent Ligand Enables NanoBRET Binding Studies and Single-Molecule Microscopy at the Histamine H3 Receptor

Abolishing Dopamine D2long/D3 Receptor Affinity of Subtype-Selective Carbamoylguanidine-Type Histamine H2 Receptor Agonists

Histamine H2 receptor radioligands: triumphs and challenges

Collaborators5

Katarzyna Szczepańska

David Reiner-Link

Enrique José Cobos Del Moral

Barry Finzel

Ulrich Gergs

How do I reach out?